Publications

SELECT: 2030 – 2026 | 2025 – 2021 | 2020 – 2016 | 2015 – 2011 | 2010 – 2006 | 2005 – 1999

(66) H. Mizoguchi, G. C. Micalizio “Synthesis of Highly Functionalized Decalins via Metallacycle-Mediated Cross-Coupling” J. Am. Chem. Soc. 2015, 137, 6624-6628.

(65) G. C. Micalizio, S. Hale “Reaction Design, Discovery, and Development as a Foundation to Function-Oriented Synthesis” Acc. Chem. Res. (invited), 2015, 48, 663-673.

(64) W. S. Kim, C. Aquino, Mizoguchi, H.; G. C. Micalizio “LiOOt-Bu as a Terminal Oxidant in a Titanium-Mediated [2+2+2] Reaction Cascade” Symposium-in-Print (invited), Tetrahedron Lett. 2015, 56, 3557-3559.

(63) X. Cheng, G. C. Micalizio “An Annulation Reaction for the Synthesis of Cross-Conjugated Triene-containing Hydroindanes from Acyclic Precursors” Org. Lett. 2014, 16, 5144-5147.

(62) V. Jeso, C. Aquino, X. Cheng, H. Mizoguchi, M. Nakashige, G. C. Micalizio “Synthesis of Angularly Substituted Trans-fused Hydroindanes by Convergent Coupling of Acyclic Precursors” J. Am. Chem. Soc. 2014, 136, 8209-8212.

(61) Comprehensive Organic Synthesis II. G. C. Micalizio “Early Transition Metal-Mediated Reductive Coupling Reactions” In: Comprehensive Organic Synthesis, 2nd edition; Gary A. Molander and Paul Knochel (eds.), Oxford: Elsevier; 2014; Vol. 5; pp. 1660-1737.

(60) X. Li, V. Jeso, S. Heyward, G. S. Walker, R. Sharma, G. C. Micalizio, M. D. Cameron, “Characterization of T-5 N-oxide Formation as the First Highly Selective Measure of CYP3A5 Activity” Drug Metabolism and Disposition, 2014, 42, 334-342.

(59) D. P. Canterbury, O. Kubo, K. N. Scott, J. L. Cleveland, G. C. Micalizio, “Synthesis of C11-Desmethoxy Soraphen A_1a: A natural product analog that inhibits acetyl-CoA carboxylase” ACS Med. Chem. Lett. 2013, 4, 1244-1248.

(58) D. Yang, G. C. Micalizio, “Stereochemical Lability of Azatitanacyclopropanes and an Efficient Dynamic Kinetic Reoslution in Reductive Cross-Coupling Reactions with Allylic Alcohols” Chem. Commun. 2013, 49, 8857-8859.

(57) V. Jeso, S. Iqbal, P. Hernandez, M. D. Cameron, H. Park, P. V. LoGrasso, G. C. Micalizio “Synthesis of Benzoquinone Ansamycin-Inspired Macrocyclic Lactams from Shikimic Acid” Angew. Chem. Int. Ed. 2013, 52, 4800-4804.

(56) V. Jeso, C. Yang, M. D. Cameron, J. L. Cleveland, G. C. Micalizio “Synthesis and Structure–Activity Relationships of Lehualide B – A Marine-derived Natural Product with Potent Anti-Multiple Myeloma Activity” ACS Chemical Biology, 2013, 8, 1241-1252.

(55) V. Jeso, G. C. Micalizio “Relay catalysis at a boron centre” Nature (News and Views) 2013, 494, 179-181.

(54) M. Sarkar, B. D. Pascal, C. Steckler, C. Aquino, G. C. Micalizio, T. Kodadek, M. J. Chalmers “Decoding Split-and-Pool Combinatorial Libraries with Electron Transfer Dissociation Tandem Mass Spectrometry” J. Am. Soc. Mass Spec. 2013, 24, 1026-1036.

(53) O. Kubo, D. P. Canterbury, G. C. Micalizio “Synthesis of the C1-C26 Hexacyclic Subunit of Pectenotoxin 2” Org. Lett. 2012, 14, 5748-5751.

(52) D. Yang, G. C. Micalizio “Synthesis of Alkaloid (–)-205B via Stereoselective Reductive Cross-Coupling and Intramolecular [3+2] Cycloaddition” J. Am. Chem. Soc. 2012, 134, 15237-15240.

(51) P. S. Diez, G. C. Micalizio “Convergent Synthesis of Deoxypropionates” Angew. Chem. Int. Ed. 2012, 51, 5152-5156.

(50) S. Greszler, H. A. Reichard, G. C. Micalizio “Asymmetric Synthesis of Dihydroindanes by Convergent Alkoxide-Directed Metallacycle-Mediated Bond Formation” J. Am. Chem. Soc. 2012, 134, 2766-2774.

(49) M. Z. Chen, G. C. Micalizio “Three-Component Coupling Sequence for the Regiospecific Synthesis of Substituted Pyridines” J. Am. Chem. Soc. 2012, 134, 1352-1356.

(48) C. Aquino, M. Sarkar, M. J. Chalmers, K. Mendez, T. Kodadek, G. C. Micalizio “A Biomimetic Polyketide-Inspired Approach to Small Molecule Ligand Discovery” Nature Chem. 2012, 4, 99-104.

(47) Science of Synthesis – Knowledge Updates 2012/4: G. C. Micalizio “Titanium-Mediated Reductive Cross-Coupling (Intermolecular Metallacycle-Mediated C–C Bond Formation)” Science of Synthesis, 2012, 33-97.

(46) D. Yang, G. C. Micalizio, “Convergent and Stereodivergent Synthesis of Complex 1-Aza-7-Oxabicyclo[2.2.1]heptanes” J. Am. Chem. Soc. 2011, 133, 9216-9219.

(45) M. A. Tarselli, K. M. Raehal, A. K. Brasher, C. Groer, M. D. Cameron, L. M. Bohn, G. C. Micalizio, “Synthesis of Conolidine, a Potent Non-Opioid Analgesic for Tonic and Persistent Pain” Nature Chem. 2011, 3, 449-453.

(44) V. Jeso, L. Cherry, T. K. Macklin, S. C. Pan, P. V. LoGrasso, G. C. Micalizio “Convergent Synthesis and Discovery of a Natural Product-Inspired Paralog-Selective Hsp90 Inhibitor” Org. Lett. 2011, 13, 5108-5111.

(43) D. P. Canterbury, G. C. Micalizio “Convergent Route to the CDEF Tetracycle of Pectenotoxin-2” Org. Lett. 2011, 13, 2384-2387.

(42) H. A. Reichard, G. C. Micalizio “Metallacycle-Mediated Cross-Coupling with Substituted and Electronically Unactivated Alkenes” Chem. Sci. 2011, 2, 573-589.

(41) D. Yang, J. K. Belardi, G. C. Micalizio “Generation of quaternary centers by reductive cross-coupling: shifting of regioselectivity in a subset of allylic alcohol-based coupling reactions” Tetrahedron Lett. 2011, 52, 2144-2147.